Payment & Shipping Terms:
|Shipping Policy:||Free Sample Available||Shipping Methods:||EMS,HKEMS,FEDEX,DHL,TNT,Aramex,ETC|
sex hormones drugs,
natural anti estrogen
Anabolic Toremifene Citrate Anti Estrogen Steroids Fareston 99% for Anti Estrogen
|Product name||Toremifene Citrate|
|Other name||FC 1157a; Fareston; NK 622; NSC 613680|
|CAS register number||89778-27-8|
|Appearance||White or almost white powder|
|Package||Discreet packing way with your choice|
|Usage||can be used as pharmaceutical material|
Toremifene Citrate Description
Toremifene Citrate (Fareston) is an anti-estrogenic medication, a SERM officially classified as a non-steroidal triphenylethylene derivative. As an anti-estrogen, Fareston functions by binding or attaching to the estrogen receptors in various tissues throughout the body creating a competition between it and the estrogen hormone. By attaching to the varying receptors this prevents the estrogen hormone from binding and performing its intended action. Primarily this will be beneficial in that it prevents the estrogen hormone from binding to the estrogen receptors in the mammary tissue.
Unlike Aromatase Inhibitors, a much stronger class of anti-estrogens, Fareston does not have the ability to lower serum estrogen levels. AI’s function by inhibiting aromatization, which refers to the conversion of testosterone to estrogen; this in turn lowers the body’s serum estrogen levels; there is now less estrogen available to do what estrogen does. However, with Fareston use, while no reduction occurs the circulating estrogen doesn’t have the ability to perform and feed breast cancer or the condition known as gynecomastia common to many steroid users.
Although anti-estrogenic in nature it is only anti-estrogenic in part. Fareston will actually act as estrogen in the liver, which will support healthier lipid profiles. As it acts as estrogen in the liver, this will support reductions in LDL cholesterol and the synthesis of HDL cholesterol. In fact, while other SERM’s carry this ability Fareston has been shown to carry it to the strongest level making it an excellent choice for the anabolic steroid user on cycle in the fight against gynecomastia.
Toremifene Citrate Application
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Licensed in the United States under the brand name Fareston, toremifene citrate is FDA-approved for use in advanced (metastatic) breast cancer. It is also being evaluated for prevention of prostate cancer under the brand name Acapodene.
It has already been covered that Toremifene is a SERM, and serves to block Estrogen at various receptor sites in certain tissues within the body (breast tissue in particular). As a layman explanation, Toremifene pretends to be a 'fake' Estrogen that occupies Estrogen receptors within breast tissue. With these receptors occupied by Toremifene, real Estrogen cannot perform their jobs there. Toremifene does not reduce total blood plasma levels of Estrogen. In addition to being antagonistic to Estrogen receptors in breast tissue, it is also antagonistic to Estrogen at the hypothalamus gland (this essentially 'tricks' the hypothalamus into thinking there is little or no circulating Estrogen levels in the body, causing it to increase its manufacture of Testosterone so that it can utilize aromatization to restore these levels.
Toremifene citrate COA
|Description||White or Almost White Crystalline Powder||White Powder|
|Loss On Drying||0.5%max||0.25%|
|Organic Volatile Impurities||meets the requirments.||Conforms|
|Residual Solvents||meets the requirments.||Conforms|
|Conclusion||The specification conform with USP32 standard|
Toremifene Citrate use/dosing
Toremifene citrate is interchangeable with tamoxifen citrate (Nolvadex) while on cycle or in post-cycle
therapy. 20mg of tamoxifen citrate = 60mg of toremifene citrate3 . From this Toremifene citrate can be extrapolated that for treatment and/or prevention of gynocomastia sixty milligrams should be sufficient for treatment. The recommended dosage for breast cancer treatment is one 60mg tablet administered once per day. During steroid treatment athletes and bodybuilders may use 30mg to 60mg per day
For use during post-cycle therapy users have anecdotally indicated that doses ranging between 60 and
120 mgs per day are average. Most users have reported when using Toremifene citrate for their post-
cycle therapy they will administer the drug for a minimum of three weeks. A maximum length has not
necessarily been established due to the few side effects associated with the compound. In this case, this
compound can be run for as long as wanted with little to no concern being needed to be paid to potential
side effects. See the below section for more details.
Female athletes occasionally use clomiphene citrate for the reduction of estrogenicity near the time of a bodybuilding contest. In some instances this may aid in increasing fat loss and muscularity, particularly in female trouble areas such as the hips and thighs. The drug, however, often produces very troubling side effects in pre-menopausal women, and is likewise not in very high demand among this group.
Related product lists
|Methenolone enanthate (Primo E)||303-42-4|
|Drostanolone Propionate (Masteron P )||521-12-0|
|Drostanolone enanthate (Masteron E)||521-12-0|
|Mixed spin Dapoxetine||129938-20-1|